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Half-life of plasmatic drug elimination (biological half-life):

a) informs, how much time will be needed for elimination of the drug from organism after discontinuation of pharmacotherapy with this drug
b) depends on the ratio (proportion) between rapidity of drug absorption and rapidity of drug elimination
c) if dosing of the drug is discontinued, after one biological half-life the concentration of the drug will have fallen to half of the initial concentration
d) informs how much time will be needed to reach the steady state of drug concentration in the case of repeated drug administration

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Final answer:

The half-life of a drug informs the time needed for its plasma concentration to decrease by half. It affects dosing frequency and can influence side effects and effectiveness. Option (b) does not describe half-life accurately, while options (a), (c), and (d) provide correct information related to drug elimination and dosing.

Step-by-step explanation:

The half-life of a drug is a crucial pharmacokinetic parameter that indicates the period of time required for the concentration of the drug in plasma to reduce to one-half of its initial value. This concept is central to understanding how often a drug should be dosed to maintain therapeutic levels without causing toxicity. Options (a), (c), and (d) are accurate descriptions of half-life in the context of drug administration. Particularly, option (a) relates to the time needed for a drug to be eliminated after treatment cessation, option (c) confirms that after one half-life the drug concentration drops to 50%, and option (d) indicates the time for drug levels to stabilize with repeated dosing. Option (b) is inaccurate since half-life is primarily determined by the rate of drug elimination independently of the rate of absorption. Understanding half-life also helps determine appropriate dosing intervals. Drugs with a short half-life may require multiple doses throughout the day to maintain efficacy, while those with longer half-lives can be dosed less frequently. For instance, a drug with a one hour half-life would likely need to be administered multiple times in a 24-hour period. Additionally, the relationship of half-life to side effects and plasma protein binding are important considerations, as these can affect not only the duration of a drug's action but also its distribution, efficacy, and toxicity.

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