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What effect does beta lactamase have on amoxicillin?

User Jerry An
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Final answer:

Beta-lactamase inactivates amoxicillin by breaking its beta-lactam ring structure, rendering it ineffective. Clavulanic acid is used to inhibit beta-lactamase and restore amoxicillin's effectiveness.

Step-by-step explanation:

Beta-lactamase is an enzyme produced by bacteria that inactivates and renders amoxicillin ineffective. Beta-lactamase breaks the beta-lactam ring structure of amoxicillin, which is essential for its antibacterial activity.

This mechanism of resistance occurs as bacteria develop the ability to produce more beta-lactamase enzymes or acquire new ones that are not inhibited by amoxicillin's beta-lactamase inhibitors. When the beta-lactamases overwhelm the inhibitory effects of the drug, the bacteria become resistant to the amoxicillin.

To combat this resistance, clavulanic acid, a beta-lactamase inhibitor, is often combined with amoxicillin in medications like Augmentin. Clavulanic acid irreversibly binds to the beta-lactamase enzymes, preventing them from inactivating the amoxicillin.

User Incognito
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