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Which of the following cholinoceptor blocking drugs is the LEAST absorbed by the brain?

1) Scopolamine
2) Ipratropium
3) Benztropine
4) Atropine

User Sotti
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1 Answer

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Final answer:

Ipratropium is the cholinoceptor blocking drug that is the least absorbed by the brain, due to its structure as a quaternary ammonium compound, limiting its ability to cross the blood-brain barrier.

Step-by-step explanation:

Out of the drugs listed, Ipratropium is the one that is the least absorbed by the brain. This is because ipratropium is a quaternary ammonium compound, which does not readily cross the blood-brain barrier. In contrast, scopolamine, benztropine, and atropine are tertiary amines that can cross the blood-brain barrier to a greater extent. Ipratropium's poor brain penetration makes it a suitable drug for respiratory treatments, such as in chronic obstructive pulmonary disease (COPD), because it minimizes systemic side effects.

User Dipak Telangre
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