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When used in place of spHM, which peptide would be most likely to achieve the same experimental results?

A. FLGFAY
B. FLGFQY
C. FLGFGY
D. FLGFEY

User Martz
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1 Answer

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Final answer:

Option B (FLGFQY) is most likely to produce results similar to SP1.7 because it retains the crucial C-terminal phenylalanine and introduces a tolerated glutamine residue in place of histidine.

Step-by-step explanation:

The question revolves around substituting the bioactive heptapeptide SP1.7 with a peptide that would most likely achieve the same experimental results. Given your options of different peptides (A-D), we must consider what modifications to H-Phe-Phe-NH₂ would retain binding affinity and improve pharmacokinetic properties while also being resistant to metabolic degradation and efflux.

Based on the information provided, which emphasizes the importance of the C-terminal phenylalanine and the potential for N-terminal modifications, option B (FLGFQY) introduces a glutamine residue in place of histidine. This switch is tolerated in similar sequences without significant loss in affinity, and the other positions remain unchanged; thus FLGFQY is most likely to produce comparable results.