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From the below list of common beta blockers, order them according to their suitability to cross membranes, taking into account their log p values?

1) Propranolol
2) Atenolol
3) Metoprolol
4) Carvedilol

User Xthexder
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Final answer:

Beta-blockers are ordered by their ability to cross membranes based on log P values, from highest to lowest: Propranolol, Carvedilol, Metoprolol, Atenolol. Log P is indicative of a drug's lipophilicity and membrane permeability.

Step-by-step explanation:

Ordering beta-blockers based on their ability to cross membranes, from highest to lowest log P values: Propranolol, Carvedilol, Metoprolol, Atenolol.

Beta-blockers are a class of medications often used to treat cardiovascular diseases by blocking beta-receptors that cause vasoconstriction and increased heart rates. The log P value is a measure of a compound's lipophilicity, or its ability to dissolve in fats, oils, and non-polar solvents. Generally speaking, a higher log P indicates better membrane permeability due to increased lipophilicity. Propranolol has a high log P value, indicating strong lipophilicity; it can readily cross cell membranes and the blood-brain barrier. Carvedilol also has a relatively high log P, meaning it's also lipophilic, though to a lesser extent compared to propranolol. Metoprolol has a lower log P value, indicating moderate membrane-crossing ability. Lastly, Atenolol, with the lowest log P among them, is less lipophilic and thus has a decreased ability to cross lipid membranes. These properties can influence the drug's distribution in the body and potential side effects profile.

User Joooeey
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