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A fall in cyclic AMP within the target cell occurs when

norepinephrine binds to which of adrenergic receptors?

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Final answer:

Norepinephrine binding to α2-adrenergic receptors causes a decrease in cyclic AMP levels within the target cell, as these receptors inhibit adenylyl cyclase through the Gi protein.

Step-by-step explanation:

A decrease in cyclic AMP (cAMP) within the target cell occurs when norepinephrine binds to α2-adrenergic receptors. The mechanism involves the α2-adrenergic receptors coupling to a G-protein known as Gi, which inhibits the action of adenylyl cyclase and thus reduces the synthesis of cAMP. Conversely, binding to β-adrenergic receptors is associated with an increase in cAMP as these receptors are coupled to Gs proteins, which stimulate adenylyl cyclase activity. Norepinephrine mainly acts through the α-adrenergic receptors, leading to a decrease in cAMP levels within the cell, which in turn can cause effects such as smooth muscle contraction.

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