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When a 500 mg dose of ampicillin was administered by bolus intravenous injection, the blood drug concentration was 10 ug/ml after 2 hours If the half ampicillin is 2 hours, calculate the -life of following: The elimination rate constant; The concentration in the blood immediately after the injection 3 The volume of distribution of ampicillin The blood concentration after 8 hours if a 1 g dose is given: The time the next dose should be given if the minimum effective concentration is 2ug/ml and 500 mg dose was given.

User Uwe Mayer
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The elimination rate constant (k) can be calculated using the following formula:

k = 0.693 / half-life

Since the half-life of ampicillin is 2 hours, the elimination rate constant can be calculated as follows:

k = 0.693 / 2 hours = 0.693 / 120 minutes = 0.0058 per minute

To calculate the concentration in the blood immediately after the injection, we can use the following formula:

C0 = C2 * e^(kt)

Where C0 is the initial concentration, C2 is the concentration after 2 hours, k is the elimination rate constant, and t is the time elapsed.

Since the initial concentration is unknown, we cannot calculate it using the above formula.

The volume of distribution (Vd) can be calculated using the following formula:

Vd = dose / C0

Since C0 is unknown, we cannot calculate the volume of distribution.

To calculate the blood concentration after 8 hours if a 1 g dose is given, we can use the following formula:

C = C0 * e^(-kt)

Where C0 is the initial concentration, k is the elimination rate constant, and t is the time elapsed.

Since the initial concentration is unknown, we cannot calculate the blood concentration after 8 hours.

To find the time the next dose should be given if the minimum effective concentration is 2ug/ml and a 500 mg dose was given, we need to determine the time it takes for the concentration to decrease to 2ug/ml.

To do this, we can use the following formula:

C = C0 * e^(-kt)

Where C0 is the initial concentration, k is the elimination rate constant, and t is the time elapsed.

We can rearrange the formula to solve for t:

t = -(1/k) * ln(C / C0)

Since C0 is unknown, we cannot calculate the time the next dose should be given.

User Jesse Jiang
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